Regioselective synthesis of 19-fluorovitamin D via fluorination of vitamin D-sulfur dioxide adducts

DOI: 10.1016/S0040-4039(96)01459-1

Source and publish data:

Tetrahedron Letters p. 6753 - 6754 (1996)

Update date:2022-07-30

Topics:

Authors:

Iwasaki, Yukiko

Shimizu, Masato

Hirosawa, Takayuki

Yamada, Sachiko

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1016/S0040-4039(96)01459-1

19-Fluorovitamin D derivatives are conveniently synthesized by the regioselective electrophilic fluorination of vitamin D-SO₂ adducts followed by defulfonylation and photochemical isomerization.

Full text of DOI:10.1016/S0040-4039(96)01459-1

Products guided by the article

Product name:(5E,7E,10Z)-3β-(tert-butyldimethylsilyloxy)-19-fluoro-9,10-seco-5,7,10(19)-cholestatriene

Cas No:182232-27-5

R&D Labs maybe for 182232-27-5

Anhui Biochem United Pharmaceutical Co., Ltd.

Contact:0086 551 5167062 / 5228268

Address:No. 30 Hongfeng Road, Hi-Tech Development Zone, Hefei (230088), China
WUHU HUAHAI BIOLOGY ENGINEERING CO LTD

Contact:+86-553-3836920

Address:7/F NO.82 LAODONG ROAD WUHU CHINA
Lyrin Industrial Corporation Limited

Contact:86-731-82571800

Address:Rm 2408,Asia Economy International Building,Shaoshan Road South,Yuhua District,Changsha,Hunan,China
Shandong Yaroma Perfumery Co., Ltd.

Contact:+86- 531- 88024598

Address:7-702 Caizhi Central, 59 Gong Ye South Road, Jinan City,250101, P. R. China
NingBO Hong Xiang Biochem.Co.Ltd

website:http://www.hxbiochem.com

Contact:0574-66003444

Address:Ning Bo Bei Lun

Relevant to this article

Doi:10.1021/jm00316a008
(1967)
Electrochemical fluorination using alkali-metal fluorides

Doi:10.1002/anie.201200438
(2012)
Novel β-iminoenolato ( or β-carbonyliminato) complexes starting from di-μ-hydroxo palladium or platinum complexes with dimethyl acetylenedicarboxylate and primary amines: Crystal structure of [NBu₄][(C₆F₅) ₂Pd{N

Doi:10.1016/0022-328X(96)06339-5
(1996)
An Efficient Protocol for a Sharpless Style Racemic Dihydroxylation

Doi:10.1016/0040-4039(95)00054-G
(1995)
2,3,18,19-Dioxidosqualene stereoisomers: characterization and activity as inhibitors of purified pig liver 2,3-oxidosqualene-lanosterol cyclase

Doi:10.1021/jo9607020
(1996)
Synthesis of 3-[1H-imidazol-4-yl] propyl 4-[¹⁸F] fluorobenzyl ether ([¹⁸F] fluoroproxyfan): A potential radioligand for imaging histamine H₃ receptors

Doi:10.1002/1099-1344(200008)43:9<873::AID-JLCR371>3.0.CO;2-A
(2000)

Article Doi