Regioselective synthesis of 19-fluorovitamin D via fluorination of vitamin D-sulfur dioxide adducts

DOI: 10.1016/S0040-4039(96)01459-1

Source and publish data:

Tetrahedron Letters p. 6753 - 6754 (1996)

Update date:2022-07-30

Topics:

Authors:

Iwasaki, Yukiko

Shimizu, Masato

Hirosawa, Takayuki

Yamada, Sachiko

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Article abstract of DOI:10.1016/S0040-4039(96)01459-1

19-Fluorovitamin D derivatives are conveniently synthesized by the regioselective electrophilic fluorination of vitamin D-SO₂ adducts followed by defulfonylation and photochemical isomerization.

Full text of DOI:10.1016/S0040-4039(96)01459-1

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