A Suzuki coupling approach to trifluoromethyl derivative of targretin (LGD 1069)

DOI: 10.1016/S0960-894X(97)00382-X

Source and publish data:

Bioorganic and Medicinal Chemistry Letters p. 2117 - 2120 (1997)

Update date:2022-08-05

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Authors:

Qing, Feng-Ling

Fan, Junfa

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Article abstract of DOI:10.1016/S0960-894X(97)00382-X

The palladium-catalyzed Suzuki coupling reaction σ-trinuoromethylated arylboronic acid 4 and vinyl triflate 5 provided the trifluoromethyl derivative of Targretin (LGD1069).

Full text of DOI:10.1016/S0960-894X(97)00382-X

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