Synthesis of Optically Active Condensed Tetrahydropyridin-3-ones as Precursors of Alkaloid Analogues

DOI: 10.1055/s-1997-1521

Source and publish data:

Synlett p. 1071 - 1072 (1997)

Update date:2022-09-26

Topics:

Authors:

Faltz, Heike

Radspieler, Alexander

Liebscher, Jürgen

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Article abstract of DOI:10.1055/s-1997-1521

Reaction of α-aminoester 2 with o-bromobenzylbromide or 3-bromo-2-bromomethylindole 1 gives N-alkylation products 3, which further undergo intramolecular acylation upon Br/Li-exchange. This sequence represents the first access to optically active condense

Full text of DOI:10.1055/s-1997-1521

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Product name:L-Alanine, N-[(2-bromophenyl)methyl]-N-(phenylsulfonyl)-, methyl ester

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