Solution phase combinatorial chemistry. Discovery of 13- and 15-membered polyazapyridinocyclophane libraries with antibacterial activity

DOI: 10.1016/S0040-4020(98)00131-8

Source and publish data:

Tetrahedron p. 3999 - 4012 (1998)

Update date:2022-08-03

Topics:

Authors:

An, Haoyun

Wang, Tingmin

Mohan, Venkatraman

Griffey, Richard H.

Dan Cook

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Article abstract of DOI:10.1016/S0040-4020(98)00131-8

A solution phase simultaneous addition of functionalities (SPSAF) combinatorial approach was utilized to synthesize 40 polyazacyclophane libraries (total complexity of 4275). Eighteen different functionality sets, utilizing 42 functionalities, were design

Full text of DOI:10.1016/S0040-4020(98)00131-8

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