Retinoid X receptor-antagonistic diazepinylbenzoic acids

DOI: 10.1248/cpb.47.1778

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1778 - 1786 (1999)

Update date:2022-08-02

Topics:

Authors:

Ebisawa, Masayuki

Umemiya, Hiroki

Ohta, Kiminori

Fukasawa, Hiroshi

Kawachi, Emiko

Christoffel, Ghislaine

Gronemeyer, Hinrich

Tsuji, Motonori

Hashimoto, Yuichi

Shudo, Koichi

Kagechika, Hiroyuki

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.47.1778

Several dibenzodiazepine derivatives were identified as novel retinoid X receptor (RXR) antagonists on the basis of inhibitory activity on retinoid- induced cell differentiation of human promyelocytic leukemia cells HL-60 and transactivation assay using r

Full text of DOI:10.1248/cpb.47.1778

NII-Electronic Library Service

Products guided by the article

Product name:4-(5,7,7,10,10-pentamethyl-7,8,9,10,12,13-hexahydro-5H-5,13-diaza-benzo[4,5]cyclohepta[1,2-b]naphthalen-12-yl)-benzoic acid methyl ester

Cas No:208171-13-5

R&D Labs maybe for 208171-13-5

hangzhou feixia327

Contact:--

Address:80G, No.1 Building, Guodu Development Mansion, No. 182 Zhaohui Road, Hangzhou City, Zhejiang Province,China.
Zhejiang kehong chemical co., ltd

Contact:0086-575-85522000

Address:xiner center RD binhai industrial zone shaoxing zhejiang province P.R.China,312073
Hangzhou JINLAN Pharm-Drugs Technology Co., Ltd

website:http://www.jlpharms.com

Contact:+86-571-86982636

Address:Rm A606, Fuyi Center, jianqiao street, Jianggan Area
Shanghai He Yang International Trading Co., Ltd.

Contact:+86-21-52043598

Address:Room 816, Blag.5, No.58 Huachi Road
Nanjing Duly Biotech Co., Ltd

website:http://www.dulynet.com/

Contact:025-84699383 -8003

Address:Room 503, Building 2, Chuangxinhui, No. 61 Wenjing Road, High-tech Development Zone, Pukou District, Nanjing City, Jiangsu Province Nanjing, Jiangsu

Relevant to this article

Ph₃P-I₂ mediated aryl esterification with a mechanistic insight

Doi:10.1016/j.tetlet.2016.03.105
(2016)
Low-temperature heat capacities and standard molar enthalpy of formation of the solid-state coordination compound trans-Cu(Ala)₂(s) (Ala = l-α-alanine)

Doi:10.1016/j.tca.2008.02.024
(2008)
Design and synthesis of π-extended resveratrol analogues and in vitro antioxidant and anti-inflammatory activity evaluation

Doi:10.3390/molecules26030646
(2021)
Doi:10.1021/jo01110a603
(1956)
Newer synthes of the pyoluteorin antibiotics.

Doi:10.1016/S0040-4039(00)99733-8
(1970)
An efficient and simple approach for the synthesis of pyranopyrazoles using imidazole (catalytic) in aqueous medium, and the vibrational spectroscopic studies on 6-amino-4-(4′-methoxyphenyl)-5-cyano-3-methyl-1-phenyl-1,4- dihydropyrano[2,3-c]pyrazole using density functional theory

Doi:10.1016/j.saa.2011.06.033
(2011)

Article Doi