Retinoid X receptor-antagonistic diazepinylbenzoic acids

DOI: 10.1248/cpb.47.1778

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 1778 - 1786 (1999)

Update date:2022-08-02

Topics:

Authors:

Ebisawa, Masayuki

Umemiya, Hiroki

Ohta, Kiminori

Fukasawa, Hiroshi

Kawachi, Emiko

Christoffel, Ghislaine

Gronemeyer, Hinrich

Tsuji, Motonori

Hashimoto, Yuichi

Shudo, Koichi

Kagechika, Hiroyuki

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.47.1778

Several dibenzodiazepine derivatives were identified as novel retinoid X receptor (RXR) antagonists on the basis of inhibitory activity on retinoid- induced cell differentiation of human promyelocytic leukemia cells HL-60 and transactivation assay using r

Full text of DOI:10.1248/cpb.47.1778

NII-Electronic Library Service

Products guided by the article

Product name:4-(5,7,7,10,10-pentamethyl-7,8,9,10,12,13-hexahydro-5H-5,13-diaza-benzo[4,5]cyclohepta[1,2-b]naphthalen-12-yl)-benzoic acid methyl ester

Cas No:208171-13-5

R&D Labs maybe for 208171-13-5

Chongqing maohuan Chemicals Co., Ltd

website:http://www.bschem.com

Contact:+86 13996103726

Address:Chongqing Nan'an District Tu Town
Zibo Ocean International Trade Co.,Ltd(expird)

Contact:+86 533 5160706

Address:1117, Hongtai Bld., Songling rd, Zichuan,Zibo,Shandong,China
Shanghai Yuking Water Soluble Material Tech Co., Ltd

Contact:86-21-68286299

Address:4F, 13B, No. 600, South Xinyuan Road 201306, Shanghai, China
Tradlon Chemical Co., Ltd.

Contact:+86-710-3516804

Address:Number 83,Panggong road,Xiangcheng District,Xiangyang ,Hubei
Jinan Trio PharmaTech Co., Ltd

Contact:86-531-88811783；+(0)13153010282

Address:2766 Yingxiu Road, Jinan High-Tech Zone, China

Relevant to this article

Ph₃P-I₂ mediated aryl esterification with a mechanistic insight

Doi:10.1016/j.tetlet.2016.03.105
(2016)
Low-temperature heat capacities and standard molar enthalpy of formation of the solid-state coordination compound trans-Cu(Ala)₂(s) (Ala = l-α-alanine)

Doi:10.1016/j.tca.2008.02.024
(2008)
Design and synthesis of π-extended resveratrol analogues and in vitro antioxidant and anti-inflammatory activity evaluation

Doi:10.3390/molecules26030646
(2021)
Doi:10.1021/jo01110a603
(1956)
Newer synthes of the pyoluteorin antibiotics.

Doi:10.1016/S0040-4039(00)99733-8
(1970)
An efficient and simple approach for the synthesis of pyranopyrazoles using imidazole (catalytic) in aqueous medium, and the vibrational spectroscopic studies on 6-amino-4-(4′-methoxyphenyl)-5-cyano-3-methyl-1-phenyl-1,4- dihydropyrano[2,3-c]pyrazole using density functional theory

Doi:10.1016/j.saa.2011.06.033
(2011)

Article Doi