Synthesis of novel proline and γ-lactam derivatives as non-peptide mimics of Somatostatin/Sandostatin

DOI: 10.1016/S0040-4020(99)00561-X

Source and publish data:

Tetrahedron p. 10135 - 10154 (1999)

Update date:2022-08-03

Topics:

Authors:

Damour, Dominique

Herman, Frederic

Labaudiniere, Richard

Pantel, Guy

Vuilhorgne, Marc

Mignani, Serge

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Article abstract of DOI:10.1016/S0040-4020(99)00561-X

Original proline or γ-lactam derivatives bearing either an aryl group such as a phenyl or a 3-indolyl in position 3 of the proline moiety or on the 3-methyl chain of the γ-lactam skeleton were prepared as non-peptide mimics of Somatostatin/Sandostatin.

Full text of DOI:10.1016/S0040-4020(99)00561-X

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