Bioorganic and medicinal chemistry letters p. 1591 - 1594 (2002)
Update date:2022-07-30
Topics: Evaluation Antagonists Discovery Text format Experimental Chemical terms N-(triazin-1,3,5-yl) phenylalanine derivatives VLA-4 integrin
Porter, John R
Archibald, Sarah C
Brown, Julien A
Childs, Kirstie
Critchley, David
Head, John C
Hutchinson, Brian
Parton, Ted A H
Robinson, Martyn K
Shock, Anthony
Warrellow, Graham J
Zomaya, Alex
SAR studies aimed at improving the rate of clearance of a series of VLA-4 integrin antagonists by the introduction of a 1,3,5-triazine as an amide isostere are described.
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(2000)Doi:10.1002/aoc.5822
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