Bioorganic and Medicinal Chemistry Letters p. 959 - 963 (2004)
Update date:2022-08-05
Topics:
Miller, John F.
Furfine, Eric S.
Hanlon, Mary H.
Hazen, Richard J.
Ray, John A.
Robinson, Laurence
Samano, Vicente
Spaltenstein, Andrew
A novel series of P1′ chain-extended arylsufonamides was synthesiszed and evaluated for wild-type HIV protease inhibitory activity and in vitro antiviral activity against wild type virus and two protease inhibitor-resistant mutant viruses. All of the comp
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