The synthesis of substituted 2-aminophenyl heterocycic ketones

Article abstract of DOI:10.1080/00397919308013295

The synthesis of substituted 2-aminophenyl heterocyclic ketones, key intermediates to the preparation of 1,4-benzodiazepines has been achieved in one step and in good, yield from the corresponding anthranilic acid, by treatment with heterocyclic lithium reagents and chlorotrimethylsilane.

Full text of DOI:10.1080/00397919308013295

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Synthetic Communications: An
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The Synthesis of Substituted
2-Aminophenyl Heterocyclic
Ketones
R. I. Fryer a , P. Zhang a & R. Rios a
a Department of Chemistry Rutgers , The State
University of New Jersey , 73 Warren Street,
Newark, NJ, 07102
Published online: 23 Sep 2006.
To cite this article: R. I. Fryer , P. Zhang & R. Rios (1993) The Synthesis of Substituted
2-Aminophenyl Heterocyclic Ketones, Synthetic Communications: An International
Journal for Rapid Communication of Synthetic Organic Chemistry, 23:7, 985-992, DOI:
10.1080/00397919308013295
To link to this article: http://dx.doi.org/10.1080/00397919308013295
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