Chemistry Letters p. 159 - 162 (1980)
Update date:2022-09-26
Topics:
Nagao, Yoshimitsu
Seno, Kaoru
Miyasaka, Tadayo
Fujita, Eiichi
A new efficient procedure for synthesis of macrocyclic amides has been exploited by aminolysis of thiazolidine-2-thione amide (1) of dicarboxylic acid with diamines (4), or spermidine (7).A variety of macrocyclic diamides (5 and 8) and/or tetramides (6, 9, 12, and 13) have been synthesized in high yields.One can monitor the reaction, since the original yellow color of the starting material (1) disappears at the end of the reaction.
View MoreShanghai AoBo Bio-Pharmaceutical Technology Co., Ltd.
Contact:+86-21-51320130-801, 816
Address:Room 601, No. 1011, Halei Road, Zhangjiang High-Tech Park, Pudong, Shanghai
Cangzhou Senary Chemical Science-tech Co., Ltd
Contact:+86-317-3563899, 3563699
Address:168 Jinde Road, Cangzhou, Hebei, China
Shanghai Balmxy Pharmaceutical Co., Ltd
Contact:0086-21-24206007
Address:Room 402, 15#, No. 909 wangyue Road, shanghai, P. R. China
Shanghai Gsyn Chemical Co.,Ltd.
Contact:86-021-67158290
Address:86-021-67158291
Contact:+86-571-86217390
Address:No.567 Dengcai Street,Sandun,Westlake District,Hangzhou310030,Zhejiang,China.
Doi:10.1039/C39730000341
(1973)Doi:10.1021/jo00182a005
(1984)Doi:10.1039/DT9900000641
(1990)Doi:10.1021/om0109105
(2002)Doi:10.1007/s11178-005-0103-4
(2004)Doi:10.1002/anie.200351465
(2003)
