Synthesis and structure-activity relationships of a series of benzazepine derivatives as 5-HT2C receptor agonists

Article abstract of DOI:10.1016/j.bmc.2007.12.009

To identify potent and selective 5-HT_2C receptor agonists, a series of novel benzazepine derivatives were synthesized, and their structure-activity relationships examined. The compounds were evaluated for their 5-HT_2C, 5-HT_2A