Structure-activity relationship studies of novel pyrazolo[1,5-c][1,3]benzoxazines: Synthesis and benzodiazepine receptor affinity

Article abstract of DOI:10.1002/ardp.19963291204

Some 2-arylpyrazolo[1,5-c][1,3]benzoxazin-5-ones 1 and 5 oxopyrazolo[1,5-c][1,3]benzoxazin-2-carboxylates 2 were prepared and biologically evaluated for their binding at benzodiazepine receptor (BZR) in rat cortical membranes. Structure-activity relations