Bioorganic and Medicinal Chemistry Letters p. 751 - 754 (2005)
Update date:2022-08-02
Topics:
Buckley, George M.
Davies, Natasha
Dyke, Hazel J.
Gilbert, Philip J.
Hannah, Duncan R.
Haughan, Alan F.
Hunt, Caroline A.
Pitt, William R.
Profit, Rachael H.
Ray, Nicholas C.
Richard, Marianna D.
Sharpe, Andrew
Taylor, Alicia J.
Whitworth, Justine M.
Williams, Sophie C.
The development of a series of novel quinazolinethiones and quinazolinediones as inhibitors of inosine monophosphate dehydrogenase (IMPDH) is described. The synthesis, in vitro inhibitory values for IMPDH II and in vitro inhibitory value for PBMC proliferation are discussed.
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