Bioorganic and Medicinal Chemistry Letters p. 751 - 754 (2005)
Update date:2022-08-02
Topics:
Buckley, George M.
Davies, Natasha
Dyke, Hazel J.
Gilbert, Philip J.
Hannah, Duncan R.
Haughan, Alan F.
Hunt, Caroline A.
Pitt, William R.
Profit, Rachael H.
Ray, Nicholas C.
Richard, Marianna D.
Sharpe, Andrew
Taylor, Alicia J.
Whitworth, Justine M.
Williams, Sophie C.
The development of a series of novel quinazolinethiones and quinazolinediones as inhibitors of inosine monophosphate dehydrogenase (IMPDH) is described. The synthesis, in vitro inhibitory values for IMPDH II and in vitro inhibitory value for PBMC proliferation are discussed.
View MoreContact:+86-571-86217390
Address:No.567 Dengcai Street,Sandun,Westlake District,Hangzhou310030,Zhejiang,China.
Anqing World Chemical Co., Ltd.
Contact:+86-556-5800026
Address:Daguan Economic Development Zone of circular economy industrial park Anqing City Anhui province
website:http://www.herbpurify.com
Contact:0086-028-85249238
Address:Room709-C1,Incubator Building, Tianfu Life Science Park No.88,Keyuan Road,Gaoxin district,Chengdu City,Sichuan Prov,China
Ji'an Hairui Natural Plant Co. Ltd.
Contact:0796-8105528
Address:Meilin industry park, Qingyuan district Ji'an City, Jiangxi Province
website:http://www.guarson.com
Contact:+86-523-88059600,+86-13805268803
Address:Room B1006,Yafang Building,Jiangyan Avenue,Jiangyan District, Taizhou City,Jiangsu,China
Doi:10.1002/adsc.200900658
(2010)Doi:10.1002/hc.21099
(2013)Doi:10.1021/ja01854a005
()Doi:10.1002/hlca.200390050
(2003)Doi:10.1021/jo0497196
(2004)Doi:10.1016/S0040-4020(01)97396-X
(1974)