Reductive amination of piperidines with aldehydes using borane-pyridine

Article abstract of DOI:10.1080/00397919308009840

Borane-pyridine complex (BAP) was found to be an excellent replacement for NaCNBH₃ in the Borch reduction. Assorted aromatic, heterocyclic and aliphatic aldehydes were reacted with various substituted piperidines using standardized conditions.

Full text of DOI:10.1080/00397919308009840

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Synthetic Communications: An
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Communication of Synthetic
Organic Chemistry
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Reductive Amination of
Piperidines with Aldehydes
Using Borane-Pyridine
Alan E. Moormann a
a Department of Chemistry, G. D. Searle & Co. ,
4901, Searle Parkway, Skokie, IL, 60077, U.S.A.
Published online: 23 Sep 2006.
To cite this article: Alan E. Moormann (1993) Reductive Amination of Piperidines with
Aldehydes Using Borane-Pyridine, Synthetic Communications: An International Journal
for Rapid Communication of Synthetic Organic Chemistry, 23:6, 789-795
To link to this article: http://dx.doi.org/10.1080/00397919308009840
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