Bioorganic and Medicinal Chemistry Letters p. 1291 - 1294 (2004)
Update date:2022-09-26
Topics:
Pissarnitski, Dmitri A.
Asberom, Theodros
Boyle, Craig D.
Chackalamannil, Samuel
Chintala, Madhu
Clader, John W.
Greenlee, William J.
Hu, Yueqing
Kurowski, Stanley
Myers, Joyce
Palamanda, Jairam
Stamford, Andrew W.
Vemulapalli, Subbarao
Wang, Yuguang
Wang, Peng
Wu, Ping
Xu, Ruo
Development of structure-activity relationship of cyclic guanines I lead us to discovery of a potent and selective series of phosphodiesterase 5 inhibitors 52-59 (IC50=1.3-11.0 nM, PDE6/5=116-600).
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Doi:10.1055/s-2003-40342
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