β-Tosylethylamine: A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams

DOI: 10.1021/jo00099a006

Source and publish data:

Journal of Organic Chemistry p. 5856 - 5857 (1994)

Update date:2022-08-05

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Authors:

DiPietro, Darren

Borzilleri, Robert M.

Weinreb, Steven M.

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Article abstract of DOI:10.1021/jo00099a006

Readily prepared β-tosylethylamine (3) can be used to synthesize N-tosylethyl (TSE)-protected amido compounds and β-lactams, which can be deprotected under mild conditions with potassium tert-butoxide.

Full text of DOI:10.1021/jo00099a006

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