SYNTHESIS OF MONO- AND DI-ACYLATED L-2,6-DIAMINO-4-HEXYNOIC ACID POTENTIAL DERIVATIVES FOR PREPARATION OF (3)H-LABELLED LYSINE CONTAINING PEPTIDES

Article abstract of DOI:10.1016/S0040-4039(00)92878-8

The selective acylation of the 6-amino group of 2,6-diamino-4-hexynoic acid was obtained in high overall yield by a simple approach instead of copper complex method.