Synthesis and analgesic properties of two leucine-enkephalin analogues containing a conformationally restrained N-terminal tyrosine residue

DOI: 10.1021/jm00359a024

Source and publish data:

Journal of Medicinal Chemistry p. 762 - 765 (1983)

Update date:2022-08-05

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Authors:

Deeks Deeks

Crooks Crooks

Waigh Waigh

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Article abstract of DOI:10.1021/jm00359a024

Two analogues of Leu-enkephalin, in which the terminal tyrosine-1 residue has been replaced by a conformationally restrained tyrosine analogue, have been synthesized by classical solution methods, and their opiate agonist potencies on electrically stimula

Full text of DOI:10.1021/jm00359a024

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