Preparation of iodine-123 labeled AM251: A potential spect radioligand for the brain cannabinoid CB1 receptor

DOI: 10.1002/(SICI)1099-1344(199610)38:10<875::AID-JLCR908>3.0.CO;2-G

Source and publish data:

Journal of labelled compounds and radiopharmaceuticals p. 875 - 881 (1996)

Update date:2022-08-03

Topics:

Authors:

Lan, Ruoxi

Gatley, S. John

Makriyannis, Alexandros

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/(SICI)1099-1344(199610)38:10<875::AID-JLCR908>3.0.CO;2-G

We report the synthesis and labeling with iodine-123 of N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole -3-carboxamide (AM251). This compound is an anlog of the recently described cannabinoid receptor antagonist, R141716A,

Full text of DOI:10.1002/(SICI)1099-1344(199610)38:10<875::AID-JLCR908>3.0.CO;2-G

Products guided by the article

Product name:Lithium, [1-(4-bromobenzoyl)-3-ethoxy-1-methyl-2,3-dioxopropyl]-

Cas No:850554-39-1

R&D Labs maybe for 850554-39-1

KA-SHING Business Trade Macau Co., Ltd.

Contact:00853-28430045

Address:23rd Floor, Block 3 La Cite, Areia Preta, Macao
Fujian Huitian Biological Pharmacy Co., Ltd.

Contact:0086-598-8300831; 8339920

Address:No.46,Taijiang Road,Sanming City,Fujian,China
Dongtai Xinyuan Chemical Co., Ltd.

Contact:+86-21-56733000

Address:404F, 99Nong No.117 Zhongtan Rd. Shanghai
Shanghai Yuking Water Soluble Material Tech Co., Ltd

Contact:86-21-68286299

Address:4F, 13B, No. 600, South Xinyuan Road 201306, Shanghai, China
HENAN NEW BLUE CHEMICAL CO.,LTD

website:http://www.newbluechem.com

Contact:86-371-55170693/55170694

Address:Zhengzhou International Trade New Territory,Jinshui District,Zhengzhou ,China

Relevant to this article

Novel trifluoromethyl sydnone derivatives: Design, synthesis and fungicidal activity

Doi:10.1016/j.bmcl.2021.128114
(2021)
Reactions with heterocyclic enamines. Synthesis of new isoxazole derivatives

Doi:10.1002/ardp.19833160204
(1983)
Isoindolo[2,1-c][2,3]benzodiazepines

Doi:10.1002/ardp.19833160205
(1983)
First enantiospecific synthesis of (+)-β-herbertenol

Doi:10.1016/j.tet.2005.01.050
(2005)
Synthesis of monomers bearing at the 2′-position cyanomethoxycarbonyl group for phosphoramidite oligonucleotide synthesis

Doi:10.1081/NCN-200026053
(2004)
In vitro characterization of salmochelin and enterobactin trilactone hydrolases IroD, IroE, and Fes

Doi:10.1021/ja0522027
(2005)

Article Doi