Journal of Medicinal Chemistry p. 4469 - 4473 (2005)
Update date:2022-08-05
Topics:
Shie, Jiun-Jie
Fang, Jim-Min
Kuo, Chih-Jung
Kuo, Tun-Hsun
Liang, Po-Huang
Huang, Hung-Jyun
Yang, Wen-Bin
Lin, Chun-Hung
Chen, Jiun-Ling
Wu, Yin-Ta
Wong, Chi-Huey
A diversified library of peptide anilides was prepared, and their inhibition activities against the SARS-CoV 3CL protease were examined by a fluorogenic tetradecapeptide substrate. The most potent inhibitor is an anilide derived from 2-chloro-4-nitroanili
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