Novel acetylcholinesterase inhibitor as increasing agent on rhythmic bladder contractions: SAR of 8-{3-[1-(3-fluorobenzyl)piperidin-4-yl]propanoyl}- 1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one (TAK-802) and related compounds

DOI: 10.1016/j.bmc.2005.01.022

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Bioorganic and Medicinal Chemistry p. 1901 - 1911 (2005)

Update date:2022-07-29

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Authors:

Ishichi, Yuji

Sasaki, Mitsuru

Setoh, Masaki

Tsukamoto, Tetsuya

Miwatashi, Seiji

Nagabukuro, Hiroshi

Okanishi, Satoshi

Imai, Shigemitsu

Saikawa, Reiko

Doi, Takayuki

Ishihara, Yuji

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Article abstract of DOI:10.1016/j.bmc.2005.01.022

As part of an on-going investigation to develop an increasing agent on rhythmic bladder contractions, 1-aryl-3-(1-benzylpiperidin-4-yl)propanones were synthesized and examined as noncarbamate acetylcholinesterase (AChE) inhibitors. Among compounds with va

Full text of DOI:10.1016/j.bmc.2005.01.022

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