Bioorganic and Medicinal Chemistry Letters p. 619 - 622 (1999)
Update date:2022-08-05
Topics:
Mederski, Werner W. K. R.
Osswald, Mathias
Dorsch, Dieter
Christadler, Maria
Schmitges, Claus-Jochen
Wilm, Claudia
The discovery, synthesis and structure-activity relationships of a series of novel benzofuro[3,2b]pyridines as non-selective endothelin ET(A)/ET(B) as well as selective ET(B) receptor antagonists are described. The most potent non-selective inhibitor 7s d
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