
Journal of Medicinal Chemistry p. 509 - 513 (1984)
Update date:2022-08-04
Topics:
Ouellet, Rene
Rousseau, Jacques
Brasseur, Nicole
Lier, Johan E. van
Diksic, Mirko
Westera, Gerrit
The reaction of ethyl chloroformate with amino compounds has been evaluated as a simple route to carbon-11 labeling of steroid hormone-receptor-based imaging agents.Both a 17β-amino analogue of estradiol and an aminoethyl derivative of the nonsteroidal es
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