Preparation of Optically Active Piperazines from Ethyl (S)-2-(2-Alkyl-1-aziridinyl)acetates

DOI: 10.1246/bcsj.59.321

Source and publish data:

Bulletin of the Chemical Society of Japan p. 321 - 322 (1986)

Update date:2022-09-26

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Authors:

Yahiro, Nobuhide

Ito, Shigekazu

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Article abstract of DOI:10.1246/bcsj.59.321

Reaction of ethyl (S)-2-(2-alkyl-1-aziridinyl)acetates with boron trifluoride etherate in a large excess of ethylamine or ammonia gives the corresponding optically active piperazines in good yields.These piperazines retain the configuration of the starting aziridines.

Full text of DOI:10.1246/bcsj.59.321

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