Human and rat monoamine oxidase-A are differentially inhibited by (S)-4-alkylthioamphetamine derivatives: Insights from molecular modeling studies

DOI: 10.1016/j.bmc.2007.05.021

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Bioorganic and Medicinal Chemistry p. 5198 - 5206 (2007)

Update date:2022-08-04

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Authors:

Fierro, Angelica

Osorio-Olivares, Mauricio

Cassels, Bruce K.

Edmondson, Dale E.

Sepulveda-Boza, Silvia

Reyes-Parada, Miguel

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Article abstract of DOI:10.1016/j.bmc.2007.05.021

Four enantiomerically pure (S)-4-alkylthioamphetamine derivatives were evaluated as monoamine oxidase (MAO) inhibitors using the human and rat isoforms of the enzyme. Molecular dockings were performed in order to gain insights regarding the binding mode o

Full text of DOI:10.1016/j.bmc.2007.05.021

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