Topographic Probes of Angiotensin and Receptor: Potent Angiotensin II Agonist Containing Diphenylalanine and Long-Acting Antagonists Containing Biphenylalanine and 2-Indan Amino Acid in Position 8

DOI: 10.1021/jm00124a028

Source and publish data:

Journal of Medicinal Chemistry p. 898 - 903 (1989)

Update date:2022-08-26

Topics:

Authors:

Hsieh, Kun-hwa

LaHann, Thomas R.

Speth, Robert C.

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Article abstract of DOI:10.1021/jm00124a028

A series of phenylalanine-mimicking amino acids with increasing conformational restraint were prepared and incorporated into angiotensin II, in order to develop topographic probes of angiotensin useful for probing receptor boundaries by molecular graphics

Full text of DOI:10.1021/jm00124a028

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