Journal of Medicinal Chemistry p. 9457 - 9472 (2016)
Update date:2022-08-18
Topics:
Doyle, Kevin
L?nn, Hans
K?ck, Helena
Van De Po?l, Amanda
Swallow, Steve
Gardiner, Philip
Connolly, Stephen
Root, James
Wikell, Cecilia
Dahl, G?ran
Stenvall, Kristina
Johannesson, Petra
A novel series of second generation DPP1 inhibitors free from aorta binding liabilities found for earlier compound series was discovered. This work culminated in the identification of compound 30 (AZD7986) as a highly potent, reversible, and selective clinical candidate for COPD, with predicted human PK properties suitable for once daily human dosing.
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