Journal of labelled compounds and radiopharmaceuticals p. 309 - 318 (1998)
Update date:2022-08-30
Topics:
Horti, Andrew G.
Koren, Andrei O.
Ravert, Hayden T.
Musachio, John L.
Mathews, William B.
London, Edythe D.
Dannals, Robert F.
The radiochemical synthesis of 2-[18F]fluoro-3-(2(S)- azetidinylmethoxy)pyridine (2-[18F]A-85380, [18F]1) was accomplished by Kryptofix 222 assisted nucleophilic no-carrier-added [18F]fluorination of 2-iodo-3-((1-tert-butoxycarbonyl-2(S)-azetidinyl)methoxy)pyridine, 2 followed by acidic deprotection. The average radiochemical yield was 10% and the average specific radioactivity was 1050 mCi/μmol, calculated at end-of- synthesis (EOS).
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