Solid-phase synthesis of dehydroalanine derivatives

Article abstract of DOI:10.1016/S0040-4039(97)10544-5

A novel solid-phase synthetic method for dehydroalanines and dehydropeptides has been developed. Elimination of the sulfone part with concomitant release from the solid support afforded the desired dehydroalanine derivatives. The products were given in good yields and excellent purities.