Boron trifluoride promoted addition of aryllithiums to estrone benzyl ether

DOI: 10.1016/S0040-4039(98)02185-6

Source and publish data:

Tetrahedron Letters p. 9427 - 9430 (1998)

Update date:2022-08-29

Topics:

Authors:

Stephan, Elie

Affergan, Thierry

Weber, Philippe

Jaouen, Gerard

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Article abstract of DOI:10.1016/S0040-4039(98)02185-6

aryllithiums did not condense with estrone benzyl ether at low temperature. The promoted addition with boron trifluoride etherate was the best method for preparing substituted 17α-arylestradiols.

Full text of DOI:10.1016/S0040-4039(98)02185-6

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