α-amidoalkylation reactions and oxidation of adducts of benzimidazoles and acyl chlorides

Article abstract of DOI:10.1080/00397919808007016

Adducts 4 of benzimidazoles and acyl chlorides were successfully used as electrophilic reagents in an intermolecular α-amidoalkylation reaction toward ketones for synthesis of 2-(2-oxoalkyl)-1,3-diacyl-2,3- dihydrobenzimidazoles 6 and oxidized with KMnO₄ to 1,3-diacyl-2,3- dihydrobenzimidazol-2-ones 7.

Full text of DOI:10.1080/00397919808007016

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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α-Amidoalkylation Reactions
and Oxidation of Adducts
of Benzimidazoles and Acyl
Chlorides
Atanas P. Venkov a & Stela Statkova-Abeghe a
a Department of Chemistry, University of Plovdiv,
Plovdiv, 4000, Bulgaria
Published online: 20 Aug 2006.
To cite this article: Atanas P. Venkov & Stela Statkova-Abeghe (1998) α-
Amidoalkylation Reactions and Oxidation of Adducts of Benzimidazoles and
Acyl Chlorides, Synthetic Communications: An International Journal for Rapid
Communication of Synthetic Organic Chemistry, 28:10, 1857-1864, DOI:
10.1080/00397919808007016
To link to this article: http://dx.doi.org/10.1080/00397919808007016
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