Practical preparation of 3-chloro-4-methoxybenzylamine hydrochloride

Article abstract of DOI:10.1080/00397910008087426

The title compound was prepared in a practical manner by chlorinating 4- methoxybenzylamine with sulfuryl chloride in acetic acid in 79-82% yields with little side reaction.

Full text of DOI:10.1080/00397910008087426

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Synthetic Communications: An
International Journal for Rapid
Communication of Synthetic
Organic Chemistry
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Practical Preparation of 3-
Chloro-4-Methoxybenzylamine
Hydrochloride
Masaki Endo a & Jim Douglas a
a Process Research, Pharmaceutical Research
Institute Bristol-Myers Squibb Candiac, Quebec,
Canada, J5R 3W3
Published online: 04 Dec 2007.
To cite this article: Masaki Endo & Jim Douglas (2000) Practical Preparation of
3-Chloro-4-Methoxybenzylamine Hydrochloride, Synthetic Communications: An
International Journal for Rapid Communication of Synthetic Organic Chemistry, 30:14,
2609-2612, DOI: 10.1080/00397910008087426
To link to this article: http://dx.doi.org/10.1080/00397910008087426
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