European Journal of Medicinal Chemistry p. 744 - 755 (2016)
Update date:2022-08-25
Topics:
Padala, Anil K.
Wani, Abubakar
Vishwakarma, Ram A.
Kumar, Ajay
Bharate, Sandip B.
N-(2,2,2-Trifluoroethyl)-N-[4-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenyl]-benzenesulfonamide (T0901317, 6) is a potent activator of pregnane-X-receptor (PXR), which is a nuclear receptor controlling P-gp expression. Herein, we aimed to inv
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