Synthetic Communications p. 2013 - 2019 (1997)
Update date:2022-08-16
Topics:
Cao, Zhisong
Camptothecin 20(S) acetate was obtained in 60% yield by reaction of camptothecin with trichloroethane in sulfuric acid. This method represents another alternative preparation of camptothecin ester using trichloroethane as acylating agent.
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