New mild and efficient synthesis of peptidosulfonamides

Article abstract of DOI:10.1080/00397910701845340

This article describes a new route to peptidosulfonamide. Our study shows how sulfinamides were first obtained via nucleophilic cleavage of 3,6-dihydrothiazine-1-oxide system and how the products can be subjected to oxidation with m-chloroperbenzoic acid