Peptide Synthesis by Prior Thiol Capture. 4. Amide Bond Formation: The Effect of Side-Chain Substituent on the Rates of Intramolecular O,N-Acyl Transfer

DOI: 10.1021/jo00367a013

Source and publish data:

Journal of Organic Chemistry p. 3320 - 3324 (1986)

Update date:2022-08-05

Topics:

Authors:

Kemp, D. S.

Galakatos, Nicholas G.

Dranginis, Stanley

Ashton, Christopher

Fotouhi, Nader

Curran, Timothy P.

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Article abstract of DOI:10.1021/jo00367a013

The effects of varying steric bulk of the side chain substituent of the acylating agent on rate of the amide bond forming step of the dibenzofuran-based thiol capture strategy were determined from rates of intramolecular isomerization of methyl S-<4-(N-be

Full text of DOI:10.1021/jo00367a013

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