Synthesis of C-2"&β- and C-2"&α-Fluoro Avermectin B1a

DOI: 10.1039/c39870000368

Source and publish data:

Journal of the Chemical Society. Chemical communications p. 368 - 370 (1987)

Update date:2022-08-05

Topics: Synthesis Yield NMR spectroscopy Catalyst Purification Reaction Conditions Reactor

Authors:

Bliard, Christophe

Escribano, Francisca Cabrera

Lukacs, Gabor

Olesker, Alain

Sarda, Pierre

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Article abstract of DOI:10.1039/c39870000368

A synthesis of protected C-2β- and C-2α-fluoro oleandrosyl fluorides is presented; coupling of these carbohydrates with avermectin B_1a monosaccharide 5-O-t-butyldimethylsilyl derivative, followed by deprotection, furnished the title compounds w

Full text of DOI:10.1039/c39870000368

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