Journal of Medicinal Chemistry p. 1929 - 1932 (1990)
Update date:2022-07-29
Topics:
Bermudez, Jose
Dabbs, Steven
Joiner, Karen A.
King, Frank D.
Indazole 1 has previously been shown to be a potent and selective 5-HT3 receptor antagonist.A novel series of potent 5-HT3 receptor antagonists, 1-indolinecarboxamides 2a-q and 1-indolecarboxamides 3b,i,j,k, is described.The activity
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