Synthesis of substituted fused pyridines, pyrazines and pyrimidines by sequential Ugi/inverse electron demand Diels-Alder transformations

DOI: 10.1016/j.tetlet.2009.07.036

Source and publish data:

Tetrahedron Letters p. 5773 - 5776 (2009)

Update date:2022-08-05

Topics:

Authors:

Akritopoulou-Zanze, Irini

Wang, Ying

Zhao, Hongyu

Djuric, Stevan W.

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Article abstract of DOI:10.1016/j.tetlet.2009.07.036

The synthesis of all four regioisomers of fused pyrrolidino-pyridines in a one-pot two-step sequential Ugi-inverse electron demand Diels-Alder reaction is described. Fused pyrrolidino-pyrazines, pyrrolidino-pyrimidines and azepinone pyridines can also be obtained in consecutive synthetic sequences.

Full text of DOI:10.1016/j.tetlet.2009.07.036

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