
Journal of Medicinal Chemistry p. 1357 - 1369 (2010)
Update date:2022-08-04
Topics:
De La Fuente, Tania
Martín-Fontecha, Mar
Sallander, Jessica
Benhamú, Bellinda
Campillo, Mercedes
Medina, Rocío A.
Pellissier, Lucie P.
Claeysen, Sylvie
Dumuis, Aline
Pardo, Leonardo
López-Rodríguez, María L.
On the basis of our previously described pharmacophore model for serotonin 5-HT6 receptor (5-HT6R) antagonists, we have designed, synthesized, and pharmacologically characterized a series of benzimidazole derivatives 1-20 that repres
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