STEREOSELECTIVE SYNTHESIS OF TILIVALLINE

DOI: 10.1016/S0040-4039(00)99602-3

Source and publish data:

Tetrahedron Letters p. 1871 - 1872 (1989)

Update date:2022-08-06

Topics:

Authors:

Nagasaka, Tatsuo

Koseki, Yuji

Hamaguchi, Fumiko

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Article abstract of DOI:10.1016/S0040-4039(00)99602-3

Tilivalline (1b) was easily synthesized by converting lactam 3b to the acyliminium precursor 5b followed by stereoselectively introducing indole from the less hindered side of 5b.

Full text of DOI:10.1016/S0040-4039(00)99602-3

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