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(1 mmol), isoxazolyl thiourea
3 (1 mmol), and ceric ammonium nitrate
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carboxylate 4a (1 mmol) and 3-amino-5-methylisoxazole 5 (1 mmol) were
heated in diphenyl ether (15 mL) at 200 °C for 10 h under N2 atmosphere. The
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reaction, the solvent was removed by vacuum distillation and the contents are
poured in ice cold water. The separated solid was filtered and recrystallized
from ethanol to give the pure product (6a–h).
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