
ACS Medicinal Chemistry Letters p. 938 - 942 (2011)
Update date:2022-08-04
Topics:
Crosignani, Stefano
Jorand-Lebrun, Catherine
Campbell, Gordon
Pretre, Adeline
Grippi-Vallotton, Tania
Quattropani, Anna
Bouscary-Desforges, Gwenaelle
Bombrun, Agnes
Missotten, Marc
Humbert, Yves
Fremaux, Christele
Paquet, Mikael
El Harkani, Kamel
Bradshaw, Charles G.
Cleva, Christophe
Abla, Nada
Daff, Hamina
Schott, Olivier
Pittet, Pierre-Andre
Arrighi, Jean-Francois
Gaudet, Marilene
Johnson, Zoe
Antagonism of the CRTH2 receptor represents a very attractive target for a variety of allergic diseases. Most CRTH2 antagonists known to date possess a carboxylic acid moiety, which is essential for binding. However, potential acid metabolites O-acyl gluc
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(2011)