The Synthesis of 1H-, 3H-, and 5H-2-Benzazepine Derivatives in the Reaction of Bicyclic Aromatic Nitro Compounds with Dimethyl Phosphite and Amines in the Basic Conditions

DOI: 10.1021/jo00003a063

Source and publish data:

Journal of Organic Chemistry p. 1283 - 1286 (1991)

Update date:2022-08-05

Topics:

Authors:

Danikiewicz, Witold

Makosza, Mieczyslaw

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Article abstract of DOI:10.1021/jo00003a063

1- and 2-nitronaphthalenes and 5-, 6-, and 8-nitroquinolines react with dimethyl phosphite and various primary and secondary amines in the presence of NaOMe in MeOH to give 1H-, 3H, and 5H-2-benzazepine or pyridazepine derivatives.Some structural features

Full text of DOI:10.1021/jo00003a063

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