2-Imino-1,3,4-thiadiazole Derivatives of GABA as GABAA Antagonists

DOI: 10.1071/CH9901767

Source and publish data:

Australian Journal of Chemistry p. 1767 - 1772 (1990)

Update date:2022-08-05

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Authors:

Allan, Robin D.

Apostopoulos, Christine

Richardson, Jennifer A.

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Article abstract of DOI:10.1071/CH9901767

New heterocyclic derivatives of GABA, with a GABA moiety on the 3 position of a 2-imino-5-aryl-1,3,4-thiadiazole ring, have been readily prepared by alkylation of 2-amino-1,3,4-thiadiazoles in dimethylformamide.They are active as GABA_A antagoni

Full text of DOI:10.1071/CH9901767

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