Journal of Medicinal Chemistry p. 2885 - 2903 (2013)
Update date:2022-08-15
Topics:
Ye, Na
Chen, Chuan-Huizi
Chen, Tiantian
Song, Zilan
He, Jin-Xue
Huan, Xia-Juan
Song, Shan-Shan
Liu, Qiufeng
Chen, Yi
Ding, Jian
Xu, Yechun
Miao, Ze-Hong
Zhang, Ao
A series of benzo[de][1,7]naphthyridin-7(8H)-ones possessing a functionalized long-chain appendage have been designed and evaluated as novel PARP1 inhibitors. The initial effort led to the first-generation PARP1 inhibitor 26 bearing a terminal phthalazin-
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