
Archiv der Pharmazie p. 803 - 806 (1993)
Update date:2022-08-05
Topics:
Kutscher
Engel
Fleischhauer
Niebch
The synthesis of four proposed metabolites 1-4 of Naftopidil, a selective α1-antagonist, is reported. These compounds comprise hydroxylated and demethylated derivatives and a cleavage product of Naftopidil.
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