Agents for the treatment of overactive detrusor. VIII. Synthesis and pharmacological properties of 4,4-diphenyl-2-cycloalkenylamines including FK584 and 3,3- or 4,4-diphenylcycloalkylamines

DOI: 10.1248/cpb.43.71

Source and publish data:

Chemical and Pharmaceutical Bulletin p. 71 - 77 (1995)

Update date:2022-08-03

Topics:

Authors:

Taniguchi

Okumura Okumura

Take Take

Tsubaki Tsubaki

Terai Terai

Nakanishi

Shiokawa

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1248/cpb.43.71

This article describes the synthesis of 4,4-diphenyl-2-cycloalkenylamines (3, 5a) including PK584 (S(-)-3a) and 3,3- or 4,4-diphenylcycloalkylamines (2, 4, 5b), and their inhibitory activities against detrusor contraction. The order of inhibitory activity

Full text of DOI:10.1248/cpb.43.71

NII-Electronic Library Service

Products guided by the article

Product name:Benzene, 1,1'-(4-azido-2-cyclopenten-1-ylidene)bis-

Cas No:138951-98-1

R&D Labs maybe for 138951-98-1

SICHUAN TONGSHENG AMINOACID CO.LTD

website:http://www.aminoacid.cc

Contact:86-838-2274206/2850606

Address:Room 1-11-1,No.19 of North TianShan Road,Deyang,Sichuan China
Sinonine Industry Co.,Ltd

Contact:86+21-56421993

Address:3F,BUILDING 10,NO.2889 JINKE ROAD, SHANGHAI.
Hangzhou Donglou Bio-nutrient Co., Ltd.

Contact:+86-571-82225795,13967112289

Address:Louta Town, Xiaoshan,Hangzhou,Zhejiang
Deer Chemicals Co., Ltd.

Contact:+86-13666670345

Address:Agricultural Development Zone, Haining, Jiaxing, Zhejiang
ANHUI CHEM-BRIGHT BIOENGINEERING CO.,LTD

Contact:86-561-4080321

Address:No.8 Lieshan Industrial Zone of Huaibei

Relevant to this article

Heterobifunctional ligands: Practical chemoenzymatic synthesis of a cell adhesive glycopeptide that interacts with both selectins and integrins

Doi:10.1021/jm000295r
(2001)
Asymmetric dihydroxylation onto the α,β-unsaturated carboxylic ester derivatives of camptothecin

Doi:10.3987/COM-97-7892
(1997)
Alkenylborane-derived frustrated Lewis pairs: Metal-free catalytic hydrogenation reactions of electron-deficient alkenes

Doi:10.1021/om3006068
(2012)
α-Amination of keto-nitrones via Multihetero-Cope rearrangement employing an imidoyl chloride reagent

Doi:10.1039/c2cc33401a
(2012)
Thermally induced [3+2] cyclization of aniline-tethered alkylidenecyclopropanes: A facile synthetic protocol of pyrrolo[1,2-a]indoles

Doi:10.1039/c2cc33269h
(2012)
An efficient synthesis of dithiocarbamates under ultrasound irradiation in water

Doi:10.1007/s00706-011-0687-z
(2012)

Article Doi