Synthesis and binding properties to GABA receptors of 3-hydroxypyridinyl- and 3-hydroxypiperidinyl-analogues of baclofen

DOI: 10.1002/ardp.19923250108

Source and publish data:

Archiv der Pharmazie p. 29 - 33 (1992)

Update date:2022-07-29

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Authors:

Desideri

Galli Galli

Sestili Sestili

Stein Stein

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Article abstract of DOI:10.1002/ardp.19923250108

The synthesis of 3-(3-hydroxy-2-pyridinyl)propanoic acid, 3-(3-hydroxy-2-pyridinyl)-4-aminobutanoic acid, their corresponding piperidine compounds, and of some cyclized derivatives is described. In vitro assays none of the new compounds shows any notewort

Full text of DOI:10.1002/ardp.19923250108

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