Synthesis and binding properties to GABA receptors of 3-hydroxypyridinyl- and 3-hydroxypiperidinyl-analogues of baclofen

DOI: 10.1002/ardp.19923250108

Source and publish data:

Archiv der Pharmazie p. 29 - 33 (1992)

Update date:2022-07-29

Topics:

Authors:

Desideri

Galli Galli

Sestili Sestili

Stein Stein

Read Full Text PDF DownLoad Join now for total 90,000,000 free articles

Article abstract of DOI:10.1002/ardp.19923250108

The synthesis of 3-(3-hydroxy-2-pyridinyl)propanoic acid, 3-(3-hydroxy-2-pyridinyl)-4-aminobutanoic acid, their corresponding piperidine compounds, and of some cyclized derivatives is described. In vitro assays none of the new compounds shows any notewort

Full text of DOI:10.1002/ardp.19923250108

Products guided by the article

Product name:2-Propenoic acid, 3-[3-(phenylmethoxy)-2-pyridinyl]-, ethyl ester, (Z)-

Cas No:139745-91-8

R&D Labs maybe for 139745-91-8

Fujian Wanke Pharmaceutical Co., LTD.

Contact:+86-598-5026002

Address:Economic development zone,jiangle county
Huayi Isotopes Co.

Contact:+ 86 512 52491118

Address:1 Fuyu Road, Haiyu TownChangshu, Jiangsu, China
Deltachem(QingDao)Co.,Ltd.

Contact:+8618766299236

Address:ROOM808, BUILDING2,NO.230 SHEN ZHEN ROAD, LAOSHAN DISTRICT
Water Chemical Co.,LTD

Contact:+86-21-6856-1349 523-87676172

Address:No16 . BinJiang Road . Taixing Economy Developing Area .JiangSu Province . China
Oren Hydrocarbons (Qingdao) Co., Ltd.

Contact:+86-532-68607667-801

Address:Room 3 # 302, No.9 Qingyun Road, Qingdao, China

Relevant to this article

An acid-catalysed hydroamination approach to isoindolines

Doi:10.1055/s-0031-1291155
(2012)
Intramolecular photoassisted cycloadditions of azaxylylenes and postphotochemical capstone modifications via suzuki coupling provide access to complex polyheterocyclic biaryls

Doi:10.1021/jo4026447
(2014)
Synthesis of homochiral 5,9-epoxybenzocyclooctenes with aminosubstituents: Relationship between structure and CNS-activity

Doi:10.1002/ardp.19933261011
(1993)
N-Protection of amines using pyridinium 2,2,2-trifluoroacetate ionic liquid as an efficient and reusable catalyst

Doi:10.1016/j.cclet.2013.11.052
(2014)
Design and synthesis of heterocyclic cations for specific DNA recognition: From AT-rich to mixed-base-pair DNA sequences

Doi:10.1021/jo402599s
(2014)
Switching enantioface selection in the asymmetric nitro-mannich reaction using single chiral bis(imidazolidine)pyridine-metal catalysts

Doi:10.1055/s-0034-1378204
(2014)

Article Doi