Synthesis of 2-(3-indolyl)-4-methylenepiperidines via intramolecular cyclization of allylsilanes

Article abstract of DOI:10.1080/00397919208055412

The synthesis of 2-(3-indolyl)-4-methylenepiperidines using an efficient formation of the piperidine ring by intramolecular reaction between an allylsilane group and an iminium ion is reported.

Full text of DOI:10.1080/00397919208055412

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Synthetic Communications: An
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Organic Chemistry
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Synthesis of 2-(3-Indolyl)-4-
Methylenepiperidines VIA
Intramolecular Cyclization of
Allylsilanes
Mario Rubiralta a , Anna Diez a , David Miguel a
Roland Remuson b & Yvonne Gelas-mialhe b
,
a Laboratory of Organic Chemistry, Faculty of
Pharmacy , University of Barcelona , 08028,
Barcelona, Spain
b Laboratoire de Chimie des Substances Naturelles ,
Universite Biaise Pascal , associe au CNRS (URA 485),
63177, Aubiere, France
Published online: 05 Dec 2006.
To cite this article: Mario Rubiralta , Anna Diez , David Miguel , Roland Remuson &
Yvonne Gelas-mialhe (1992) Synthesis of 2-(3-Indolyl)-4-Methylenepiperidines VIA
Intramolecular Cyclization of Allylsilanes, Synthetic Communications: An International
Journal for Rapid Communication of Synthetic Organic Chemistry, 22:3, 359-367, DOI:
10.1080/00397919208055412
To link to this article: http://dx.doi.org/10.1080/00397919208055412
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